http://rdf.ncbi.nlm.nih.gov/pubchem/patent/SU-1456432-A1
Outgoing Links
Predicate | Object |
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assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_ca5f07e41553d5ad03b10dad0242c158 http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_9d3ebd367c63b9d9acd12ea1aaee215b http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_7da89c7b38c555fd425cd6bb45a95da3 http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_560a26364f29956460d47b5868ac9ea1 http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_69919ba572f6e8dfba00f61256a44fdd |
classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D403-04 |
filingDate | 1987-07-23-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
grantDate | 1989-02-07-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c17b4544cc6dd939ff13f8f66378e959 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1d37d8f930672715ffa0eebb75637676 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c93968294eb0d3b6a17faa6252a317fa http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_04508e1fe91d87d330d8053248faf6c2 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_903243f07a44a9f657b1d441d9275084 |
publicationDate | 1989-02-07-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber | SU-1456432-A1 |
titleOfInvention | Method of producing (1-acetylpyrazolidinyl-5)indols |
abstract | The invention relates to heterocyclic compounds, in particular, a process for the preparation of (1-acetylpyrazolidinyl-5) indoles of the general formula CH3C C9-N-CH-X-CH2-CHR / t-N-. where X is CeH t-n-Rs, a group of the formula R, 73E-ir VR. R and R - H or OH., F J 4 5 LP OI l RI - H, CHj or CHj-CjHy, which can be used as intermediate products for the synthesis of biologically active substances. The goal is to create new intermediates for the synthesis of new active substances. Synthesis of the target compounds is carried out by the reaction of the indole of the general formula HX, where X is as above, and 1-acetyl-5-oxypyrazoline is of the general formula CH3C0-K-CH OH - € Nn-CH "L - Y-SbH1 -P -P5 "where R4 and R - see above, in the presence of an ion-exchange resin Ku-2 in H®-form in an inert organic solvent medium. Output%, t.sh1., C, gross formula: a) 15; 184-186; CaflH.NjO; b) 82; 114-115; C., E..N.O: c) 80; 186-188; Ci.HjsNjO; d) 91, - 210-212; .NjO; e) 27; 225-226; , The method allows to synthesize new compounds of the pyrazolidinidol series, which cannot be obtained by other methods. 2 S (L |
priorityDate | 1987-07-23-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 38.