http://rdf.ncbi.nlm.nih.gov/pubchem/patent/SK-5897-A3
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_c7ad58d3c0b071069a8ee0cb8c8ba2e8 |
| classificationCPCAdditional | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/Y02P20-55 |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D413-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P31-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D215-38 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-47 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P31-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D221-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-435 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-42 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D263-18 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-41 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D413-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D215-38 |
| filingDate | 1997-01-15-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_80befe1826b529ea5d5fc3178a59a425 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_52b096a566d89b5fb8cb6facfb2660b2 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_63c0fd119ffe9d8bb6f1b71fe12065a1 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_4148d0476ad139d275222faac1b98fbc http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c66d142f62c574f729030855d8675ac2 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_f901b24a2225435183659b50b5763168 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_38c126a42b2a9626a9462f568dde2218 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_8497726e35c9068fa4f1b9a4a44caccc |
| publicationDate | 1997-09-10-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | SK-5897-A3 |
| titleOfInvention | 2-oxo and 2-thio-1,2-dihydroquinolinyl-oxazolidinones, method for producing them, their use and pharmaceutical composition containing same |
| abstract | 2-(Oxo or thio)-1,2-dihydroquinolinyl-oxazolidinones (I) and their isomers and salts are new: A = O or S; D = H; 3-6C cycloalkyl; alkoxycarbonyl with up to 4C; alkyl or alkenyl with up to 9C optionally substituted by CN, CF3, halo, OH, pyridyl, Ph, COOH, CONH2, alkoxycarbonyl with up to 5C, naphthyl, 3-6C cycloalkyl and/or -(CO)a-NR<2>R<3>, -N(R<4>)-SO2-R<5>, -SO2-N-R<6>R<7> or -S(O)b-R<8>; acyl with up to 5C optionally substituted by CF3, CCl3 or OR<9>; -(CT)d-NR<10>R<11>; -(CO)e-NR<12>-CO-NR<13>R<14>; -NR<15>-SO2R<16>R<17>R<18>-N-SO2-; R<19>-S(O)f; or -CO-R<20>; E, L = H; COOH; halo; CN; CHO; CF3; NO2; or 1-4C alkyl; R<1> = N3; OH; OR<21>; OSO2R<22>; or NR<23>R<24>; a, d, e = 0 or 1; f, b = 0-2; R<2>-R<4>, R<6>, R<7> = H; 1-5C alkyl; or Ph; or NR<2>R<3> = morpholinyl, thiomorpholino, pyrrolidinyl, piperazinyl or piperidyl optionally substituted on a free N atom by alkyl or acyl with up to 4C; R<5>, R<8> = 1-6C alkyl, Ph; benzyl; or tolyl; R<9> = H or 1-5C alkyl optionally substituted by Ph or naphthyl; T = O or S; R<10>-R<15>, R<17>, R<18> = as R<2>-R<4>; R<16>, R<19> = = R<5> and R<8>; R<20> = 6-10C aryl optionally substituted by halo; R<21> = acyl with up to 6C or a OH protecting group; R<22> = 1-5C alkyl; Ph; or toluoyl; R<23>, R<24> = H; 3-6C cycloalkyl; Ph; 1-6C alkoxy; t-Boc; Fmoc; benzyloxycarbonyl; 1-6C alkyl optionally substituted by CN or alkoxycarbonyl with up to 4C; -CT-R<25>; P(O)(OR<26>)(OR<27>) or -SO2-R<28>; R<25> = H; 3-6C cycloalkyl; CF3; 1-6C alkoxy; Ph; Ph-CH2O; 1-6C alkyl optionally substituted by alkoxycarbonyl with up to 5C, CN, F, Cl, Br or CF3; thioalkyl or acyl with up to 5C; or -NR<29>R<30>; R<26>, R<27> = H or 1-4C alkyl; R<28> = 1-4C alkyl or Ph; and R<29>, R<30> = H; Ph; or 1-4C alkyl. |
| priorityDate | 1996-01-16-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 200.