http://rdf.ncbi.nlm.nih.gov/pubchem/patent/SK-279820-B6

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filingDate 1993-06-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_b416faa126310dc84ef80e5f790e2c6b
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_a1547556ce020ce3d89a3f87227a3a8a
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publicationDate 1999-04-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber SK-279820-B6
titleOfInvention PHARMACEUTICAL PREPARATION FOR LOCAL USE, SPÔSO
abstract A pharmaceutical composition for topical administration, comprising asymmetric lamellar aggregates, comprising phospholipids having a phosphatidylcholine content of 30 to 99 percent by weight, pharmacological active compounds and fluorocarbon, the amount of fluorocarbon being in the range from 1 to 100 percent by weight/volume, in a pharmaceutical excipient suitable for topical administration. A process for the preparation of a phospholipid-containing pharmaceutical composition comprising the steps of emulsifying phospholipids having a phosphatidylcholine content of 30 to 99 percent by weight with a fluorocarbon or fluorocarbon mixture, a pharmacological active compound or an active compound combination being incorporated into the emulsion, and the amount of fluorocarbon being in the range from 1 to 100 percent by weight/volume to produce asymmetric lamellar aggregates; and incorporating the asymmetric lamellar aggregates obtained in this way into an excipient suitable for topical administration as active compound carriers having a particle size from 50 nm to 1000 nm. The pharmaceutical composition and use thereof in the preparation of ointments, creams, lotions, pastes, gels, powders or a dressing or plaster or sprays.
priorityDate 1992-06-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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