http://rdf.ncbi.nlm.nih.gov/pubchem/patent/SG-11201403216U-A
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filingDate | 2013-02-14-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_7f158de296769b519637c3e44a5fe0bb http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_645b9cc46912ae7c349bc9c0aef98990 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_b80cc72f5171aca22ec47b90fdf1d231 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_83080f2d4f59bfb2deef3b6c4e41bf9f http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_a5559847434048a77f451260c10203b1 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_6801b90cc3638bb86fb6262d6344ef3d http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1cc7a62df961f2b7348dee000e6d6742 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_a5c99336886d00cd2a4ad685905044ea http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_996e4357043a929e36ca0d44fad69e21 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_4b1b6decd35fadc0765345d4fe900491 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_312879328270785fbacf38177f538f63 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_6d262cf44e97d6f3d732b9583c8c98b3 |
publicationDate | 2014-12-30-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber | SG-11201403216U-A |
titleOfInvention | Methods and compounds useful in the synthesis of orexin-2 receptor antagonists |
abstract | (12) INTERNATIONAL APPLICATION PUBLISHED UNDER THE PATENT COOPERATION TREATY (PCT) (19) World Intellectual Property Organization International Bureau (43) International Publication Date 22 August 2013 (22.08.2013) WIPOIPCT (10) International Publication Number WO 2013/123240 A1 (51) International Patent Classification: C07C 29/147 ( 2006.01) C07C 303/28 (2006.01) C07D 239/28 (2006.01) C12P 41/00 (2006.01) C07C 33/50 (2006.01) C07C 309/70 (2006.01) C07D 239/34 (2006.01) C07D 401/12 (2006.01) (21) International Application Number: PCT/US2013/026204 (22) International Filing Date: (25) Filing Language: (26) Publication Language: 14 February 2013 (14.02.2013) English English (30) Priority Data: 61/600,109 17 February 2012 (17.02.2012) US (71) Applicant: EISAI R&D MANAGEMENT CO., LTD [JP/JP]; 6-10 Koishikawa, 4-Chome Bunkyo-ku, Tokyo, 112-8088 (JP). (72) Inventors; and (71) Applicants (for US only): MONIZ, George, Anthony [US/US]; 700 Huron Avenue, Apt. 18K, Cambridge, MA 02138 (US). WILCOXEN, Annie, Zhu [US/US]; 18 Peter Road, North Reading, MA 01864 (US). BENAYOUD, Farid [US/US]; 805 Forest Streeet, North Andover, MA 01845 (US). LEE, Jaemoon [KR/US]; 57 Argilla Road, Andover, MA 01810 (US). ZHANG, Huiming [CN/US]; 2 Dorset Circle, Andover, MA 01810 (US). TERAUCHI, Taro [JP/JP]; c/o Eisai Co., Ltd. Tsukuba Research, Labor atories 1-3 Tokodai 5-chome, Tsukuba-shi, lbaraki (JP). TAKEMURA, Ayumi [JP/JP]; c/o Eisai Co., Ltd. Tsukuba Research, Laboratories 1-3 Tokodai 5-chome, Tsukuba-shi, lbaraki (JP). YOSHIDA, Yu [JP/JP]; c/o Eisai Co., Ltd. Tsukuba Research, Laboratories 1-3 Tokodai 5-chome, Tsukuba-shi, lbaraki (JP). TANAKA, Toshiaki [JP/JP]; c/o Eisai Co., Ltd. Tsukuba Research, Laboratories 1-3 Tokodai 5-chome, Tsukuba-shi, lbaraki (JP). SORIMACHI, Keiichi [JP/JP]; c/o Eisai Co., Ltd. Tsukuba Research, Laboratories 1-3 Tokodai 5-chome, Tsukuba-shi, lbara (JP). NAOE, Yoshimitsu [JP/JP]; c/o Eisai Co., Ltd. Tsukuba Research, Laboratories 1-3 Tokodai 5-chome, Tsukuba-shi, lbaraki (JP). KAZUTA, Yuji [JP/JP]; c/o Eisai Co., Ltd. Tsukuba Research, Labor atories 1-3 Tokodai 5-chome, Tsukuba-shi, lbaraki (JP). (74) Agent: MYERS BIGEL SIBLEY & SAJOVEC, P.A.; P.O. Box 37428, Raleigh, NC 27627 (US). (81) Designated States (unless otherwise indicated, for every kind of national protection available)'. AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW. (84) Designated States (unless otherwise indicated, for every kind of regional protection available)'. ARIPO (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, SZ, TZ, UG, ZM, ZW), Eurasian (AM, AZ, BY, KG, KZ, RU, TJ, TM), European (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR), OAPI (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG). Published: — with international search report (Art. 21(3)) © •t CJ m CJ i-H o CJ (54) Title: METHODS AND COMPOUNDS USEFUL IN THE SYNTHESIS OF OREXIN-2 RECEPTOR ANTAGONISTS 5 (57) Abstract: The present disclosure provides compounds and methods that are useful for the preparation of compounds useful as orexin-2 receptor antagonists. |
priorityDate | 2012-02-17-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
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isDiscussedBy | http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID56841936 http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID451203623 |
Total number of triples: 49.