http://rdf.ncbi.nlm.nih.gov/pubchem/patent/RU-2753335-C2

Outgoing Links

Predicate Object
assignee http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_3d7e2f8fb5650d7d3616661464b67771
classificationCPCAdditional http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07B2200-13
classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P5-50
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-4035
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P3-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P3-10
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P3-12
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D405-04
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P35-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D309-14
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P3-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-4035
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P5-50
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D405-04
filingDate 2017-08-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2021-08-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_007de1921d00622e48a511dcb89305e8
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_eeb1bef21626a7e7a93fbbf86de0b253
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c9d8e18f1998f1a4ef62e59b5ebe64a6
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_283bbe2adefd647d30b545c3f294aabb
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_f96748adfa511ea43f81bdb976019afe
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_7c5c634975ef17b315f112e57b39dae8
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_f060ce97a6c1a4391989682dad1dad8b
publicationDate 2021-08-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber RU-2753335-C2
titleOfInvention Long-acting dpp-iv inhibitor crystal and its salts
abstract FIELD: chemistry. n SUBSTANCE: invention relates to a crystal of compound (2R,3S,5R) - 5-(5-methanesulfonylisoindoline-2-yl) - 2-(2,5-difluorophenyl)tetrahydro-2H-pyran-3-amine, represented by the formula (I). The invention also relates to the phosphate of the compound of formula (I), with a molar ratio of the compound of formula (I) to orthophosphoric acid equal to 1:1, to the fumarate of the compound of formula (I), with a molar ratio of the compound of formula (I) to fumaric acid equal to 1:0.5, as well as to the phosphate and fumarate crystals of the compound of formula (I). n EFFECT: compounds of the invention are intended as a long acting DPP-IV inhibitor. n n n n 15 cl, 11 dwg, 8 tbl, 11 ex
priorityDate 2016-08-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

Incoming Links

Predicate Subject
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2016127916-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2007097931-A2
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EA-018613-B1
isDiscussedBy http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9833925
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID2641
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID429192758
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID396196
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID25253
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID54678486
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419554785
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID1061
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID46209133
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID723
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID132229448
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419538597
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID411550719
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID411550722
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419533737
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421239439
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID397492
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5885
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID3772480
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415744028
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID429192686
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID45031
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID455667478
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4946
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID1004
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5462311
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID565888
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID132229437
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122493962
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419546881
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID83717
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID424920351
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID69797
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122493960
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419567032
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1803
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID3772194
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID280802
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID450749712
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415777671
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID397595
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426213184
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID3771769
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11721
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100301982
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2733271
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID444972
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID12629
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID14795871
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419474096
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID281122
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID494052
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID452561397
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID14526
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID16102683
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID13482
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID450796724
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID451875064
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421381364
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID373686
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID414871259
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10703

Total number of triples: 95.