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filingDate 2018-06-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2019-05-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_506ae7a89eb7841d1e144456a3ff38bb
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publicationDate 2019-05-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber RU-2688235-C1
titleOfInvention Pharmaceutical anti-diabetic composition based on substituted thiophene carboxylate and a method for production thereof
abstract FIELD: medicine; pharmaceuticals. n SUBSTANCE: group of inventions refers to medicine, chemical-pharmaceutical industry and pharmacy, more specifically to a pharmaceutical composition for oral administration, having hypoglycemic and hypolipidemic activity. Pharmaceutical composition contains (Z)-ethyl 2-(4-(4-chlorophenyl)-2,4-dioxo-3-(3-oxo-3,4-dihydroquinoxalin-2(1H)-ylidene)butanamido)-4-methyl-5-phenylthiophene-3-carboxylate as an active substance and additives –microcrystalline cellulose, sodium croscarmellose, crospovidone, lactose monohydrate, partially pregelatinized corn starch, stearic acid salt. Pharmaceutical composition is presented in the form of a tablet coated with a coating. Second invention relates to a method for preparing a pharmaceutical composition which consists in using wet granulation and direct pressing of various components. n EFFECT: group of inventions is characterized by sufficient mechanical strength, high therapeutic activity, satisfactory technological characteristics and stable during storage for at least 2 years. n 12 cl, 1 tbl, 3 ex
priorityDate 2018-06-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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