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publicationDate 2017-10-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber RU-2633061-C2
titleOfInvention Neprilysin inhibitors
abstract FIELD: veterinary medicine. n SUBSTANCE: preparation for external and local application is applied pointwise or by watering. Pets are cats or dogs. The composition contains an effective amount of 4-[5-(3,5-dichlorophenyl)-5-trifluoromethyl-4,5-dihydroisoxazol-3-yl]-2-methyl-N-[(2,2,2-trifluoroethylcarbamoyl)methyl]benzamide of compound (A) in a veterinarily acceptable liquid carrier. The liquid carrier contains N,N-diethyl-3-methylbenzamide in a mixture of at least two of the following solvents: acetone, ethyl-L-lactate, dimethylsulfoxide, dimethylacetamide and glycofurol, as well as an effective amount of macrocyclic lactone compound and/or insect growth-regulating compound. n EFFECT: good drug penetration in topical application and preservation of an acceptable cosmetic look of the animal. n 9 cl, 4 tbl, 7 dwg, 8 ex
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