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grantDate 2015-12-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2015-12-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber RU-2570198-C2
titleOfInvention SALTS AND POLYMORPHS OF 8-FLUORO-2-{4-[(METHYLAMINO)METHYL]PHENYL}-1,3,4,5-TETRAHYDRO-6H-AZEPINO[5,4,3-cd]INDOL-6-ONE
abstract FIELD: chemistry. n SUBSTANCE: invention relates to camsilate and maleate salts of 8-fluoro-2-{4-[(methylamino)methyl]phenyl}-1,3,4,5-tetrahydro-6H-azepino[5,4,3-cd]indol-6-one and to a pharmaceutical composition having activity which is mediated by poly(ADP-ribose)polymerase (PARP), which contains a therapeutically effective amount of the disclosed salt. n EFFECT: obtaining camsilate and maleate salts of 8-fluoro-2-{4-[(methylamino)methyl]phenyl}-1,3,4,5-tetrahydro-6H-azepino[5,4,3-cd]indol-6-one, having high hydration resistance. n 15 cl, 38 dwg, 31 tbl, 31 ex
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