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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-4375
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D471-06
filingDate 2010-01-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2011-09-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_d340d957385d3aa3181f43a63c07e821
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_51e7c4f419ee9b2c5761804e08d6ceb6
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publicationDate 2011-09-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber RU-2429840-C1
titleOfInvention Agent preventing mammal normal cell transformation in malignant cells
abstract FIELD: medicine. n SUBSTANCE: group of inventions refers to substances preventing malignant regeneration of mammal (including human) normal cells in malignant cells. Aaptos sp. sponge is used to produce an aaptamine analogue, namely 3-N-morpholinyl-9-demethyloxyaaptamine exhibiting ability to prevent mammal normal cell transformation in malignant cells. What is offered is use of 3-N-morpholinyl-9-demethyloxyaaptamine, and also its analogues 9-demethyloxyaaptamine, isoaaptamine, 3-phenethylamino-9-demethyl oxyaaptamine and 3-isopentyl amino-9-demethyloxyaaptamine as such agent. Besides, these substances are used for preparing pharmaceutical compositions preventing mammal normal cell transformation in malignant cells. 3-N-morpholinyl-9-demethyloxyaaptamine and its analogues have a cancer-preventive effect in the concentration nontoxic for normal cells. n EFFECT: reduced risk of toxic action on body after prolonged administration of the substances. n 3 cl, 1 dwg, 10 tbl, 7 ex
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-112500409-A
priorityDate 2010-01-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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