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publicationDate 2011-04-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber RU-2415840-C2
titleOfInvention 3,5-substituted piperidines as renin inhibitors
abstract FIELD: medicine, pharmaceutics. n SUBSTANCE: there are described 3,4-substituted piperidines applicable in diagnostics and drug therapy of a warm-blooded animal, preferentially for therapy of a disease which depends on renin activity; application of a compound of such kind for preparing a pharmaceutical composition for therapy of the disease which depends on renin activity; application of the compound of such kind for therapy of the disease which depends on renin activity; the pharmaceutical compositions containing 3,4-substituted piperidine, and/or a therapeutic mode involving administration of 3,4-substituted piperidine, a method for producing 3,4-substituted piperidine. The preferential compound (which also can be presented in the form of salts) are described by formula I' wherein R1, R2, T, R3 and R4 are such as described by the patent claim. n EFFECT: production of the compounds for therapy of the disease which depends on renin activity. n 28 cl, 1 tbl, 375 ex
priorityDate 2005-12-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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