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filingDate 2004-01-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2008-08-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_ce7c39a4b1d0521f149b342ac0a5ba6a
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publicationDate 2008-08-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber RU-2330849-C2
titleOfInvention MALONAMIDE DERIVATIVES AS γ-SECRETASE INHIBITORS
abstract FIELD: chemistry. n SUBSTANCE: invention concerns malonamide derivatives of the formulae (IA) or (IB) , and pharmaceutically acceptable acid additive salts of them, where R 1 , R 1 ',(R 2 ) 1,2,3 , R 3 , R 4 , R 14 , L, and are such as described in this invention. Also the invention concerns a medicine with inhibition effect on γ-secretase, which can be applied in treatment of Alzheimer's disease. n EFFECT: obtaining new malonamide derivatives with beneficial biological properties. n 17 cl, 188 ex
priorityDate 2003-02-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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