http://rdf.ncbi.nlm.nih.gov/pubchem/patent/RU-2278117-C2
Outgoing Links
| Predicate | Object |
|---|---|
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D413-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D487-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P31-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D471-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P31-04 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-4162 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-422 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-519 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D413-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D487-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D471-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D498-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P31-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-437 |
| filingDate | 2000-08-02-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| grantDate | 2006-06-20-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_5d101d78da70285faed1154a8a217c93 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_d7be3cb2b19cc77ab6471efaa94274d9 |
| publicationDate | 2006-06-20-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | RU-2278117-C2 |
| titleOfInvention | Antibacterial heterobicyclic substituted phenyloxazolidinones |
| abstract | FIELD: organic chemistry, medicine. n SUBSTANCE: invention relates to bicyclic heterocyclic substituted phenyloxazolidinones that represent compounds of the formula (I): wherein R is taken from the group consisting of -OH, O-heteroaryl, -N 3 , -OSO 2 R'', -NR'''R'''', or the formula: wherein: (ii) R'' represents direct or branched alkyl comprising up to 5 carbon atoms; (iii) R''' and R'''' are taken independently from the group consisting of hydrogen atom (H), -CO 2 -R 1 , -CO-R 1 , -CS-R 1 and -SO 2 -R 4 wherein R 1 is taken among the group consisting of cycloalkyl comprising from 3 to 6 carbon atoms and direct or branched alkyl comprising up to 6 carbon atoms; R 4 is taken from direct or branched alkyl comprising up to 4 carbon atoms; and R 4a represents -CN or -NO 2 ; R 4b represents -SR 4c , amino-group, -NHR 4c or -NR 4c R 4d wherein R 4c and R 4d are taken independently from hydrogen atom (H) or alkyl; X represents from 0 to 4 members taken independently from the group consisting of halogen atom; and Y represents radical of the formula (II): or (III): wherein R 5 , R 6 , R 7 and R 8 represent independently hydrogen atom (H), or R and R 6 and/or R 7 and R 8 form in common oxo-group; R 9 and R 10 represent independently hydrogen atom (H); A, B, C and D are taken from carbon atom (C) and nitrogen atom (N) to form phenyl ring or 5-6-membered heteroaromatic ring wherein the indicated heteroaromatic ring comprises from 1 to 4 members taken from the group consisting of nitrogen atom (N); Z is taken from alkyl, heteroaryl comprising nitrogen atom (N); and m represents 0 or 1. These compounds are useful as antibacterial agents and can be used for treatment of patient with the state caused the bacterial infection or with the bacterial infection caused by S. aureus and E. faecium . n EFFECT: valuable medicinal properties of compounds. n 45 cl, 1 tbl, 50 ex |
| isCitedBy | http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-9988406-B2 http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-10065947-B1 http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-10913752-B2 http://rdf.ncbi.nlm.nih.gov/pubchem/patent/RU-2556234-C2 http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-9328087-B2 http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-9624250-B2 http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-10702527-B2 http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-10442829-B2 http://rdf.ncbi.nlm.nih.gov/pubchem/patent/RU-2659792-C1 |
| priorityDate | 1999-08-12-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 204.