http://rdf.ncbi.nlm.nih.gov/pubchem/patent/RU-2121344-C1

Outgoing Links

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assignee http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_8be5467238d2f02d35f1fcbe430ecdaf
classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K9-48
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K9-4808
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K9-4858
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K47-12
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K47-12
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K9-48
filingDate 1991-10-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 1998-11-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_be01c737886305830d40784c8f30ff97
publicationDate 1998-11-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber RU-2121344-C1
titleOfInvention Medicinal form of biphase effect exhibiting releasing for lipophilic preparations and a method of its preparing
abstract FIELD: medicine, pharmacy. SUBSTANCE: medicinal form is used by oral route and consists of two phases: phase of nonprolonged releasing and phase of prolonged releasing the components. Form has C 12 -C 24 -fatty acid and pharmaceutically active lipophilic substance. Phase of nonprolonged releasing has part of fatty acid and phase of prolonged releasing has the rest part of fatty acid and at least part of pharmaceutically active substance. Mass ratio of fatty acid and an active substance is from 10:1 to 1:1. C 12 -C 24 -fatty acid is an oleic and/or linolenic acid. Pharmaceutically active lipophilic substance is a propranolol, verapamil, nifedipin, diltiazem, methoprolol, nicardipine and/or labetolol. New medicinal form promotes an absorption redistribution of drug from portal circulatory system to lymphatic system and excludes drug metabolism at its the first passing through the liver. Drug bioavailability is enhanced. EFFECT: enhanced effectiveness of medicinal form. 13 cl, 2 ex
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/RU-2457821-C2
priorityDate 1990-10-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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