http://rdf.ncbi.nlm.nih.gov/pubchem/patent/RU-2015108894-A
Outgoing Links
| Predicate | Object |
|---|---|
| classificationCPCAdditional | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/Y02A50-30 |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D417-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D413-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D413-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D409-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D405-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D405-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D403-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D403-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D401-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D401-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P19-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P17-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P11-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P1-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-416 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-404 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-5377 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D209-26 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P5-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P43-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D231-56 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P37-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P37-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P37-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-4439 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-437 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P29-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D471-04 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-5377 |
| filingDate | 2013-08-14-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationDate | 2016-10-10-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | RU-2015108894-A |
| titleOfInvention | COMPOUNDS OF 4-HETEROARYL SUBSTITUTED BENZOIC ACID AS RORGAMMAT INHIBITORS AND THEIR APPLICATIONS |
| abstract | 1. The compound according to formula I: or a pharmaceutically acceptable salt or solvate thereof, wherein: Y is CH, CR or N; N is 0, 1, 2, 3 or 4; A is CR or N, A is CR or N, A is CR or N, A is CR or N, provided that no more than two of the A-A can be N; R is (C) alkyl or (C) cycloalkyl; R is: (i) (C) carbocyclyl (C) alkyl; (ii) a 4-12 membered heterocyclyl (C) alkyl or (iii) (C) alkoxy, each optionally substituted with one, two, three, four or five R; R is a guide roxycarbonyl, hydroxycarbonyl (C) alkyl, (C) alkylsulfoxyaminocarbonyl or carbamoyl; R is hydrogen, halogen, cyano, nitro, hydroxy, (C) alkylcarbonyloxy, (C) alkylsulfonylamino, (C) alkylcarbonylamino, (C) alkylamino, alkyl, hydroxyl (C) alkyl or (C) alkoxy, where (C) alkyl and (C) alkoxy are optionally substituted with one or more halogens; R-R are independently hydrogen, halogen, amino, cyano, hydroxy, (C) alkoxy, (C) alkyl, (C) alkylaminocarbonyl, (C) alkyloxycarbonylamino, (di) (C) alkylaminocarbonyl, (C) alkylcarbonylamino, (C) alkylamino, and mino (C) alkyl or formaldehyde, where (C) alkoxy, (C) alkyl, (C) alkyl) aminocarbonyl, (di) (C) alkylaminocarbonyl, (C) alkylamino and amino (C) alkyl are optionally substituted with one or more halogens , hydroxyl or (C) alkoxy; or a group of the formula optionally substituted by one or more of the following: (C) alkyl, halogen, amino, cyano, hydroxy, (C) alkoxy, and where m is 1, 2, 3 or 4; R is: (i) (C) ) cycloalkyl or (C) heterocycloalkyl, both optionally substituted with one or more groups selected from halogen, amino, amino (C) alkyl, cyano, nitro, hydroxyl, oxo (= O), HNC (O), (C) alkoxycarbonyl, (di) (C) alkylaminocarbonyl, (C) alkyl or (C) alkoxy, where (C) alkoxycarbonyl, |
| priorityDate | 2012-08-15-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 286.