http://rdf.ncbi.nlm.nih.gov/pubchem/patent/RU-2014131950-A
Outgoing Links
| Predicate | Object |
|---|---|
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D413-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P33-00 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D413-10 |
| filingDate | 2013-01-29-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationDate | 2016-03-27-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | RU-2014131950-A |
| titleOfInvention | METHOD FOR PRODUCING CHARAL ISOXIDOLES OF AZETIDINE DERIVATIVES AS ANTI-PARASITIC AGENTS |
| abstract | 1. The method of obtaining the compounds of formula (1) where R, R and R each independently mean hydrogen, halo or CC-haloalkyl; R is hydroxyl or fluoro; R is CC-alkyl, C-C-alkenyl, C-C-alkyl-C-Cycloalkyl, C-C -alkylphenyl, C--C--alkylheteroaryl or C--Cг-alkylheterocycle; wherein Rоз is C--C или or C--C алки-alkyl-C-cycloalkyl, which may be optionally and independently substituted with at least one substituent selected from cyano, halo, hydroxyl , oxo, CC-alkoxy, CC-haloalkoxy, C-C-haloalkyl, -S (O) R, -SH, -S (O) NRR, -NRR, -NRC (O) R, -SC (O) R , -SCN or -C (O) NRR, and CC-alkylC-Cycloalkyl may be optionally ADDITIONAL substituted C-C-alkyl or hydroxyC-C alkilom-; where R 1 is C 1-6 alkylphenyl, C 1-6 alkylheteroaryl or C 2-6 alkylheterocycle, which may be optionally substituted with at least one substituent selected from cyano, halo, oxo, = S, hydroxyl, CC-alkoxy, C- C-alkyl, C-C-haloalkyl, -SH, -S (O) R and CC-haloalkoxy; R is C-C-alkyl or C-Cycloalkyl optionally substituted with at least one halosubstituent; R is hydrogen, CC-alkyl, or Ci-Ci-Ci-Cycloalkyl; where alkyl and alkylcycloalkyl is optionally substituted with cyano or at least one halosubstituent; R is hydrogen, C-C-alkyl, C-Cycloalkyl, C-C-alkylphenyl, C-C-alkylheteroaryl or C-C-alkylheterocycle, each of which is optionally substituted where chemically possible with at least one substituent selected from hydroxyl, cyano, halo or —S (O) R; R is CC-alkyl, C-C-haloalkyl, C-C-haloalkyl-C-cycloalkyl, C-C-alkyl -Cycloalkyl, C-C-alkylphenyl, C-C-alkylheteroaryl or C-C-alkylheterocycle, each of which is optional flaxly substituted with at least one substituent selected from cyano, halo, hydroxyl, oxo, CC-alkoxy, CC-haloalkoxy, CC-haloalkyl, -S (O) R, -SH, -S (O) NRR, -NRR, -NRC (O) R, -SC (O) R, -SCN or -C (O) NRR; n is an integer |
| priorityDate | 2012-02-03-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
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