http://rdf.ncbi.nlm.nih.gov/pubchem/patent/RU-2014127143-A
Outgoing Links
Predicate | Object |
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classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P11-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D211-34 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P11-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D211-18 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P37-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D211-20 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P11-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D211-96 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-451 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D401-12 |
classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D211-18 |
filingDate | 2012-12-10-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationDate | 2016-02-10-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber | RU-2014127143-A |
titleOfInvention | PIPERIDINYL NAPTILUXE ACIDS |
abstract | 1. The compound of formula (I): where: X is —SO— or —C (O) -; R is halogen; R is - phenyl, unsubstituted or mono - or di-substituted independently with lower alkyl, halogen, alkoxy, - SO-lower alkyl or haloalkyl, - unsubstituted heteroaryl, - lower alkyl, unsubstituted or substituted by unsubstituted phenyl or phenyl substituted by halogen, NO or NH, - unsubstituted cycloalkyl, - unsubstituted heterocycloalkyl, or - NH-phenyl, said phenyl is unsubstituted or substituted by halogen lower alkyl, haloalkyl, SO-lower alkyl or alko B; and R is lower alkyl or hydrogen, or pharmaceutically acceptable salts thereof. 2. The compound of claim 1, wherein X is —SO — .3. The compound of claim 1, wherein X is —C (O) -. 4. A compound according to claim 1, wherein R is fluorine. 5. The compound of claim 1, wherein X is —SO— and R is phenyl, unsubstituted or mono- or di-substituted independently with lower alkyl, halogen, alkoxy, —SO-lower alkyl, or —CF; unsubstituted heteroaryl; or lower alkyl unsubstituted or substituted by unsubstituted phenyl or phenyl substituted by halogen, NO or NH.6. The compound of claim 1, wherein X is —SO— and R is unsubstituted cycloalkyl; unsubstituted heterocycloalkyl; or NH-phenyl, said phenyl is unsubstituted or substituted with halogen, lower alkyl, haloalkyl, -SO-lower alkyl or alkoxy. 7. A compound according to claim 1, wherein R1 is phenyl, methylphenyl, chlorophenyl, methanesulfonylphenyl, dichlorophenyl, difluorophenyl, trifluoromethylphenyl, bis-trifluoromethylphenyl, methoxyphenyl, nitrophenyl or aminophenyl. A compound according to claim 1, wherein R4 is pyridinyl. The compound of claim 1, wherein R1 is methyl or methyl substituted with phenyl, chlorophenyl, nitroph |
priorityDate | 2011-12-12-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 94.