http://rdf.ncbi.nlm.nih.gov/pubchem/patent/RU-2012104633-A
Outgoing Links
| Predicate | Object |
|---|---|
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P1-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D207-273 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P19-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P3-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P3-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P3-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D207-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P13-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D403-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D403-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P27-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P17-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P29-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P11-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P11-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P37-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P11-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P37-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P43-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-00 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P37-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-496 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P11-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P9-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P9-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P25-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P3-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P3-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P3-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P29-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P19-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D403-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P17-00 |
| filingDate | 2010-06-11-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationDate | 2013-11-20-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | RU-2012104633-A |
| titleOfInvention | PIPERAZINYL-3-AMINOPYROLRODINE DERIVATIVES AS AN CCON2 ANTAGONIST |
| abstract | 1. A compound having the following formula I Formula 1 Formula 2 Formula 3 and Formula 4 in which: R may be independently selected from the groups consisting of a hydrogen atom, C-Cialkyl, phenyl, benzyl, benzoyl, benzenesulfonyl, C-Ci-alkylcarbonyl, C-Ci-cycloalkyl, formula II, III and IV; R, R, and R can be independently selected from the groups consisting of a hydrogen atom, C-C1-6 alkyl, phenyl and benzyl; all benzyl groups included as part of R may have many substituents independently selected from the groups consisting of C-C1-6 alkyl, C- C haloalkyl, halogen atom and cyano; R, R, R, R, R, R, R and R l are independently selected from a hydrogen atom and C-C 1-6 alkyl; R and R, R and R may be independently selected as a carbonyl group; wherein said halogen is selected from groups consisting of a fluorine, chlorine and bromine atom. 2. The compound according to claim 1, wherein the compound is selected from the groups consisting of N - {[1- (2- (1- (phenylaminocarbonyl) piperazin-4-yl) ethyl) pyrrolidine- (3R) -alkarbamoyl] methyl} -3-trifluoromethylbenzamide , N - {[1- (2- (1- (p-tolylaminocarbonyl) piperazin-4-yl) ethyl) pyrrolidin- (3R) -alkarbamoyl] methyl} -3-trifluoromethylbenzamide, N - {[1- (2- (1- (4-chlorophenylaminocarbonyl) piperazin-4-yl) ethyl) pyrrolidin- (3R) -carbamoyl] methyl} -3-trifluoromethylbenzamide, N - {[1- (2- (1- (methoxycarbonyl) piperazin-4- il) ethyl) pyrrolidin- (3R) -alkarbamoyl] methyl} -3-trifluoromethylbenzamide, N - {[1- (2- (1- (ethoxycarbonyl) piperazin-4-yl) ethyl) pyrrolidin- (3R) -yl arbamoyl] methyl} -3-trifluoromethylbenzamide, N - {[1- (2- (4-benzoylpiperazin-1-yl) ethyl) pyrrolidine- (3R) -alkarbamoyl] methyl} -3-trifluoromethylbenzamide, N - {[1- (2- (4- (2-methylbenzoyl) piperazin-1-yl) ethyl) pyrrolidin- (3R) -carbamoyl] methyl} -3-trifluoromethylbenzamide, N - {[1- (2- (4- (3-methylbenzoyl) ) piperazin-1-yl) ethyl) pyrrolidin- (3R) -carbamoyl] methyl} -3-trifluoromethylbenzamide, N - {[1- (2- (4- (4-methylbenzoyl) pi |
| priorityDate | 2009-07-10-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 63.