http://rdf.ncbi.nlm.nih.gov/pubchem/patent/RU-2010148534-A
Outgoing Links
| Predicate | Object |
|---|---|
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P27-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P3-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D471-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D487-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P3-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P3-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P3-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D498-04 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D471-04 |
| filingDate | 2009-04-21-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationDate | 2012-06-10-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | RU-2010148534-A |
| titleOfInvention | IMIDAZOLIDINONE DERIVATIVES AS INHIBITORS IN 11B-HSD1 |
| abstract | 1. Compounds of the formula:! ! where R1 represents! a) bornyl, norbornyl, bicyclo [2.2.2] octanyl or adamantyl, where bornyl, norbornyl, bicyclo [2.2.2] octanyl or adamantyl are substituted with one or two substituents independently selected from hydroxy, alkoxy, halogen, alkyl, hydroxyalkyl, amino , aminocarbonyl, alkoxycarbonyl, hydroxycarbonyl, alkylcarbonylamino groups, alkyl-S (O) 2-, alkyl-S (O) 2-amino groups, haloalkyl-S (O) 2-amino groups, alkoxycarbonylamino-S (O) 2-amino groups, amino S (O) 2-amino groups,! hydroxyalkylcarbonylamino groups, aminocarbonylamino groups, haloalkoxy groups; and where A represents CR5R6 or carbonyl; ! or b) phenyl, phenylalkyl, substituted phenyl or substituted phenylalkyl, wherein substituted phenyl and substituted phenylalkyl are substituted with one or two substituents independently selected from alkyl, halogen, haloalkyl, alkoxy, hydroxy and haloalkoxy; and where A represents CR5R6 and none of R9, R10, R11 and R12 represents a hydroxy group and R13 and R14 do not represent hydrogen simultaneously; ! R2 and R3 together with the nitrogen atom N * and the carbon atom C * to which they are attached form a group B, C, D, E, F or G:! ! ; ! R4 represents hydrogen, alkyl, cycloalkyl, cycloalkylalkyl, alkoxyalkyl, arylalkyl, arylalkoxy, hydroxyalkyl, aryl, heteroarylalkyl, heteroaryloxyalkyl, substituted aryl, substituted heteroarylalkyl, substituted heteroalkyl, substituted heteroaryl, substituted independently selected from alkyl, cycloalkyl, cyano, halogen, gal |
| priorityDate | 2008-04-30-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 116.