http://rdf.ncbi.nlm.nih.gov/pubchem/patent/RU-2010115260-A
Outgoing Links
| Predicate | Object |
|---|---|
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P1-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D491-048 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D487-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P5-50 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P7-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P7-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P3-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P3-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P3-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P3-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-28 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P27-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P27-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P3-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D413-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D417-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P43-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D413-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P13-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P15-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P15-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P17-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P17-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D401-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D401-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P19-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P19-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P19-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P19-10 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D401-10 |
| filingDate | 2008-09-03-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationDate | 2011-10-27-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | RU-2010115260-A |
| titleOfInvention | COMPOUNDS AND COMPOSITIONS AS GPR119 ACTIVITY MODULATORS |
| abstract | 1. The compound of formula I! ! wherein ! Q is a divalent or trivalent radical selected from C6-10aryl, C1-10heteroaryl, C3-8cycloalkyl and C3-8heterocycloalkyl; wherein said aryl, heteroaryl, cycloalkyl or heterocycloalkyl in Q is optionally substituted up to 3 times by radicals independently selected from halogen, C1-6 alkyl, halogen-substituted C1-6 alkyl, C1-6 alkoxy, halogen-substituted C1-6 alkoxy, -C (O) R20 and -C (O) OR20; where R20 is selected from hydrogen and C1-6 alkyl; and optionally linking a carbon atom adjacent to W2 via CR31, O, S or NR31 to a carbon atom Q to form a 5-membered ring fused to rings A and Q; where R31 is selected from hydrogen and C1-6 alkyl; ! W1 and W2 are independently selected from CR21 and N; where R21 is selected from hydrogen, cyano, C1-6 alkyl, and —C (O) OR25; where R25 is selected from hydrogen and C1-6 alkyl; ring A may contain up to 2 ring carbon atoms substituted with a group selected from —C (O) -, —C (S) - and —C (= NOR30) - and may be partially unsaturated containing up to 2 double bonds; where R30 is selected from hydrogen and C1-6 alkyl; ! L is selected from C1-6 alkylene, C2-6 alkenylene, - (CH2) nO-, -OC (O) (CH2) n-, -C (O) O (CH2) n-, -NR26 (CH2) n- and - O (CH2) n-; where R26 is selected from hydrogen and C1-6 alkyl; and n is selected from 0, 1, 2, 3, 4, and 5; where any alkyl in L may optionally be substituted with 1-3 radicals independently selected from halogen, C1-6 alkyl, halogen-substituted C1-6 alkyl, C1-6 alkoxy, halogen-substituted C1-6 alkoxy, -C (O) R22 and - C ( O) OR22; where R22 is selected from hydrogen and C1-6 alkyl; ! m is selected from 0, 1, 2, 3, and 4; ! q is selected from 0, 1, 2, 3, and 4; ! t1, t2, t3 and t4 are each independently selected from 0, 1 and 2; ! R1 is selected from -X1S (O) 0-2X2R6a, -X1S (O) 0-2X2OR6a, X1S (O) 0-2X2C (O) R6a, -1S (O) 0-2X2C (O) OR6a, -X1S (O ) 0-2X2OC (O) R6a and -X1S (O) 0-2NR6aR6b; where X1 is selected from a bond, O, NR7aR7b and C1-4 alkylene; X2 is selected and |
| priorityDate | 2007-09-20-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 194.