http://rdf.ncbi.nlm.nih.gov/pubchem/patent/RU-2010102229-A
Outgoing Links
| Predicate | Object |
|---|---|
| classificationCPCAdditional | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/Y02P20-55 |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P13-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P7-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P7-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P7-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D405-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P43-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07F9-5535 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D223-16 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P7-10 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D223-16 |
| filingDate | 2008-06-26-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationDate | 2011-08-10-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | RU-2010102229-A |
| titleOfInvention | Benzazepine derivatives suitable for use as antagonists of vasopressin |
| abstract | 1. The benzazepine compound represented by the general formula (1)! ! in which R1 denotes a group from (1-1) to (1-7):! (1-1) represents a group -CO- (CH2) n-COR2, in which n is an integer from 1 to 4, R2 is a (2-1) hydroxyl group; (2-2) a lower alkoxy group optionally substituted with a hydroxyl group, a lower alkanoyl group, a lower alkanoyloxy group, a lower alkoxycarbonyloxy group, a cycloalkyloxycarbonyloxy group or 5-methyl-2-oxo-1,3-dioxol-4-yl; or (2-3) an amino group optionally substituted with hydroxy lower alkyl; ! (1-2) represents a group -CO- (CH2) m-NR3R4 in which m is an integer from 0 to 4, R3 is a hydrogen atom or a lower alkyl group, R4- (4-1) is a hydrogen atom; (4-2) a lower alkyl group, optionally substituted with a halogen atom, a lower alkylamino group, a lower alkoxycarbonyl group or 5-methyl-2-oxo-1,3-dioxol-4-yl; or (4-3) a lower alkoxycarbonyl group optionally substituted with a halogen atom, a lower alkanoyloxy group or 5-methyl-2-oxo-1,3-dioxol-4-yl, R3 and R4 may form a 5-6 membered a saturated heterocyclic ring by linking R3 and R4 to each other, together with a nitrogen atom to which R3 and R4 are bonded directly or via a nitrogen atom or an oxygen atom, the heterocyclic ring being optionally substituted with a (4-4) lower alkyl group, if necessary substituted with hydroxy lower alkoxy; (4-5) lower alkoxycarbonyl group; (4-6) an alkylcarbonyl group (optionally substituted on the alkyl group with a carboxyl group or a lower alkoxycarbonyl group); (4-7) an arylcarbonyl group; or (4-8) boil |
| priorityDate | 2007-06-26-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 36.