http://rdf.ncbi.nlm.nih.gov/pubchem/patent/RU-2009149856-A
Outgoing Links
| Predicate | Object |
|---|---|
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D498-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P35-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P15-18 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P7-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P17-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P5-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P43-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P19-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D513-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P5-24 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P21-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-554 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P19-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P15-00 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D498-04 |
| filingDate | 2008-05-06-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationDate | 2011-06-20-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | RU-2009149856-A |
| titleOfInvention | NEW PROGRESTERON RECEPTOR MODULATORS |
| abstract | 1. (Cis) -dibenzo [b, f] l-pyrido [1,2-d] oxazepin-2-amine or (cis) -dibenzo [b, f] pyrido [1,2-d] thiazepin-2-amine according to formula I! ! where! R1 is selected from the group consisting of (1-5C) acyl, (1-5C) thioacyl, (1-4C) alkylsulfonyl and (1-4C) alkoxycarbonyl, each of which is optionally substituted with one or more halogen atoms; and! each R2 and R3 are independently selected from the group consisting of H, halogen, cyano, nitro or thiocarbamyl; and! each R4 and R5 is independently selected from the group consisting of H, (1-4C) alkyl and (1-4C) alkoxy; and! X is selected from the group consisting of -O-, -S-, -SO-, and -SO2-; ! with the proviso that when R2 is Cl, R5 is not H or its racemate. ! 2. The compound according to claim 1, characterized in that R1 represents COCH3. ! 3. The compound according to claim 1, characterized in that R1 represents COCF3. ! 4. The compound according to any one of claims 1 to 3, characterized in that R2 represents H.! 5. The compound according to any one of claims 1 to 3, characterized in that R2 represents Cl. ! 6. The compound according to any one of claims 1 to 3, characterized in that R2 is F.! 7. The compound according to any one of claims 1 to 3, characterized in that R3 represents CN. ! 8. The compound according to any one of claims 1 to 3, characterized in that R5 is methyl. ! 9. The compound according to any one of claims 1 to 3, characterized in that R5 represents a methoxy group. ! 10. The compound according to any one of claims 1 to 3, characterized in that X represents O.! 11. The compound of claim 10, wherein R1 is COCF3, R2 is H, R3 is CN, R4 is H, and R5 is CH3. ! 12. The compound of claim 10, in which R1 represents COCF3, R2 represents H, R3 represents CN, R4 represents� |
| priorityDate | 2007-05-07-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 33.