http://rdf.ncbi.nlm.nih.gov/pubchem/patent/RU-2009129119-A
Outgoing Links
| Predicate | Object |
|---|---|
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P43-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D513-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P13-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D401-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D401-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P21-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D409-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P21-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D405-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-16 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P21-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P27-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P29-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-28 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P27-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D491-048 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P35-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P35-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P31-18 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D493-04 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D401-04 |
| filingDate | 2007-12-28-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationDate | 2011-02-10-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | RU-2009129119-A |
| titleOfInvention | CARBOXAMIDE COMPOUNDS AND THEIR APPLICATION AS CALPAIN INHIBITORS |
| abstract | 1. The carboxamide compound of formula I! ! where R1 is hydrogen, C1-C10-alkyl, C2-C10-alkenyl, C2-C10-alkynyl, where the last 3 radicals mentioned may be partially or fully halogenated and / or have 1, 2 or 3 substituents R1a,! C3-C7-cycloalkyl, C3-C7-cycloalkyl-C1-C4-alkyl, where the CH2 group in the cycloalkyl fragment of the last two radicals mentioned can be substituted by O, NH, or S, or two adjacent C atoms can form a double bond, where cycloalkyl the fragment may additionally have 1, 2, 3 or 4 radicals R1b,! aryl, hetaryl, aryl-C1-C6-alkyl, aryl-C2-C6-alkenyl, hetaryl-C1-C4-alkyl or hetaryl-C2-C6-alkenyl, where aryl and hetaryl in the last 6 radicals may be unsubstituted or have 1, 2, 3 or 4 identical or different radicals R1c; ! where R1a is independently selected from OH, SH, COOH, CN, OCH2COOH, C1-C6 alkoxy, C1-C6 haloalkoxy, C3-C7 cycloalkyloxy, C1-C6 alkylthio, C1-C6 haloalkylthio, COORa1, CONRa2Ra3, SO2NRa2Ra3, -NRa2-SO2-Ra4, NRa2-CO-Ra5, SO2-Ra4, NRa6Ra7,! R1b are independently selected from OH, SH, COOH, CN, OCH2COOH, halogen, phenyl, which optionally has 1, 2 or 3 substituents R1d, or C1-C6-alkyl, C1-C6-alkoxy, C1-C6 -alkylthio where the alkyl moieties in the last 3 mentioned substituents can be partially or fully halogenated and / or have 1, 2 or 3 substituents R1a,! COORb1, CONRb2Rb3, SO2NRb2Rb3, NRb2-SO2-Rb4, NRb2-CO-Rb5, SO2-Rb4, NRb6Rb7, where,! in addition, two R1b radicals can together form a C1-C4 alkylene group, or 2 R1b radicals bonded to adjacent C cycloalkyl atoms can form together with the carbon atoms to which they are bonded, also a benzene ring,! R1c are independently selected from OH, SH, halogen, NO2, NH2, CN, CF3, CHF2, CH2F, O-CF3, O-CHF2, O-CH2F, COOH, OCH2COOH, C1-C6-alkyl, C1-C6 alkoxy, C1-C6-al |
| priorityDate | 2006-12-29-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 93.