http://rdf.ncbi.nlm.nih.gov/pubchem/patent/RU-2008129873-A
Outgoing Links
| Predicate | Object |
|---|---|
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P1-18 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P1-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P1-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P1-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-519 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P5-28 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P7-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P5-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P35-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P35-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P3-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P3-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P3-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P3-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-28 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P29-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P3-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-22 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-16 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D487-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P19-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P19-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P13-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P13-12 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D487-04 |
| filingDate | 2006-12-20-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationDate | 2010-01-27-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | RU-2008129873-A |
| titleOfInvention | CONDENSED HETEROCYCLIC COMPOUNDS USEFUL AS DPP-IV INHIBITORS |
| abstract | 1. The compound of formula (I):! ! where X represents —CH = and Y represents = N—; or X represents —C (O) - and Y represents —N (R3) -; ! R1, R2 and R3 each independently represents hydrogen, —W-hydrocarbon or —W-heterocyclyl, any of which is optionally substituted, especially in the hydrocarbon or heterocyclyl part, 1, 2, 3, 4 or 5 of R12; where one or each W independently represents a bond or linker containing from 1 to 8 atoms in the chain, and selected, for example, from -CH2-, -O-, -C (O) -, -S (O) m-, -NRa-, cyclopropylene; C1, C2, C3, C4, C5 or C6 alkyl; and their chemically appropriate combinations; and where one or each Ra is independently hydrogen, hydroxy or hydrocarbon optionally interrupted by —O— or —NH— bonds; ! R4 represents hydrogen or an electron withdrawing group, for example —CF3, —CN, —C (O) OR8, —C (O) NR8R9, —S (O) mR8 or —CH2OR10; ! R5 represents a group of formula (i):! ! where where Q is a bond or alkylene containing 1, 2 or 3 carbon atoms in a chain, optionally substituted with 1, 2, 3, 4 or 5 R12; and! Rw, Rx, Ry and Rz each independently represents hydrogen or C1-6 alkyl optionally substituted with 1, 2, 3, 4 or 5 R12; ! or two Rw, Rx, Ry, and Rz together form an alkylene bridge containing 1, 2, 3, 4, 5, or 6 carbon atoms in a chain, the bridge being optionally substituted with 1, 2, 3, 4, or 5 R12; and the other two each represents hydrogen or C 1-6 alkyl optionally substituted with 1, 2, 3, 4 or 5 R12; ! R8 and R9 are each independently hydrogen or C1-6 alkyl optionally substituted with 1, 2, 3, 4 or 5 R12; or R8 and R9, together with the nitrogen atom to which they are attached, form heterocyclyl, optionally substituted with 1, 2, 3, 4 or 5 R12; ! R10 is C1-6alkyl, C2-6alkenyl or C2-6alkynyl, any |
| priorityDate | 2005-12-23-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 167.