http://rdf.ncbi.nlm.nih.gov/pubchem/patent/RU-2008129656-A
Outgoing Links
| Predicate | Object |
|---|---|
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D401-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D401-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D405-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D409-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P43-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D413-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-28 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-30 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-16 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-18 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-22 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-24 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D401-12 |
| filingDate | 2006-12-18-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationDate | 2010-01-27-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | RU-2008129656-A |
| titleOfInvention | SUBSTITUTED PYRAZINONE DERIVATIVES AS AN ALPHA-2C-ADRENORECEPTOR ANTAGONISTS |
| abstract | 1. The compound of General formula (I)! ! its pharmaceutically acceptable acid or base addition salt, its stereochemically isomeric form, its N-oxide form or its quaternary ammonium salt, where! V represents a naphthyl radical, wherein one CH unit in the naphthyl moiety may optionally be substituted with an N atom; ! Y is a divalent radical of formula (II)! ! where a represents a nitrogen atom or carbon; ! m is an integer equal to zero, 1 or 2; ! R4 is selected from the group consisting of hydrogen, alkyl, and phenylcarboxylalkyl; ! R5 is selected from the group consisting of hydrogen and halogen; ! X1, X2 are each, independently of one another, a covalent bond, a saturated or unsaturated (C1-8) -hydrocarbon radical in which one or more divalent -CH2 units and / or one or more monovalent CH3 units may optionally be replaced by the corresponding divalent or monovalent phenyl units and in which one or more hydrogen atoms can be replaced by radicals selected from the group consisting of oxo, (C1-3) alkyloxy; halogen, cyano, nitro, formyl, hydroxy, amino, trifluoromethyl, mono- and di ((C1-3) alkyl) amino, carboxy and thio; ! p, q are, each independently from each other, an integer equal to 1 or 2; ! Q1, Q2 are, each independently of one another, a radical selected from the group consisting of hydrogen, —NR1R2, Pir, —OR3 and Het, where two —OR3 radicals can be taken together to form the divalent radical —O— (CH2 ) rO-, where r is an integer equal to 1, 2 or 3; ! R1 and R2 are, each independently of one another, a radical selected from |
| priorityDate | 2005-12-21-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
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