| abstract |
1. The compounds of formula I! ! wherein ! R1 represents Hal, OH, OA, SH, SA, H or A,! R2, R3 each, independently of each other, is -O- (X) sQ, -S- (X) sQ, -NHCO- (X) sQ, -CONH- (X) sQ, -CONA- (X) sQ, -NH (CO) NH- (X) sQ, -NH (CO) O- (X) sQ, -NHSO2- (X) sQ, -SO2NH- (X) sQ, -SO2NA- (X) sQ, NHCOA, Hal, Het or H,! where, if R2 = Н, then R3 ≠ Н, or! if R3 = H, then R2 ≠ H,! R4, R5 each, independently of one another, is H, Hal, CN, NO2, A, OH, OA, SH, SA, (CH2) nCOOH, (CH2) nCOOA, O (CH2) oCONH2, CONHA, CONAA ' , NH2, NHA, NAA ', NHCOOA, NHCO (CH2) nNH2, NHCONHA, SOA, SO2A, SO2NH2, SO2NHA, SO2NAA' or O (CH2) oHet1,! two adjacent radicals selected from the group R1, R2, R3,! together also represent methylenedioxy or ethylenedioxy,! A, A 'each, independently of each other, is a straight or branched alkyl containing 1-10 carbon atoms, in which 1-5 hydrogen atoms can be replaced by F, Cl and / or Br,! Alk or cyclic alkyl containing 3-7 carbon atoms,! A and A 'together also represent an alkylene chain containing 2-6 carbon atoms, in which one or two CH2 groups can be replaced by O, S, SO, SO2, NH, NA and / or N-COOA,! Alk is an alkenyl containing 2-6 carbon atoms,! X is a straight or branched C1-C10 alkylene or C2-C10 alkenylene, each of which is unsubstituted or mono-, two-, tri- or tetra-substituted A, OA, OH, SH, SA, Hal, NO2, CN, Ar, OAr , COOH, COOA, CHO, C (= O) A, C (= O) Ar, SO2A, CONH2, SO2NH2, CONHA, CONAA ', SO2NHA, SO2NAA', NH2, NHA, NAA ', OCONH2, OCONHA, OCONAA' , NHCOA, NHCOOA, NACOOA, NHSO2OA, NASO2OA, NHCONH2, NACONH2, NHCONHA, NACONHA, NHCONAA ', NACONAA' and / or = O, and in which one, two or three groups C can be replaced by O, S, SO, SO2 , NHCO, NACO, CONH, CONA, SO2NH, SO2NA, NHSO2, NASO2 and / or NH groups,! Q represents H, Carb, Ar or Het,! Carb is cycloalkyl containing 3-7 carbon atoms, or cycloalkenyl containing 3-7 carbon atoms, each of which is unsubstituted and |