http://rdf.ncbi.nlm.nih.gov/pubchem/patent/RS-53669-B1
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_966a6c1f382ec9bcb5e3839dfd73e5b8 |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P15-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P13-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P15-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P1-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-5517 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-22 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-24 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-18 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P29-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P1-16 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D487-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-00 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P25-22 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P25-18 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D487-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P9-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P15-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-5517 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P25-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P9-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P1-16 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P9-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P25-24 |
| filingDate | 2011-05-09-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_9f811184bcd368b898cfc7aaf03ea193 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_3fa292408c19a9787409f0a5c3d7ff9e |
| publicationDate | 2015-04-30-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | RS-53669-B1 |
| titleOfInvention | Heteroaryl-cyclohexyl-tetraaza-benzo [e] azulene |
| abstract | A compound of formula I wherein R 1 is selected from the group consisting of: i) H, ii) - C 1-6 alkyl, unsubstituted or substituted with 1 to 5 substituents individually selected from the group consisting of: OH, halogen, cyano and C 1-6 alkoxy , iii) -S (O) 2- C 1-6 alkyl, wherein C 1-6 alkyl is unsubstituted or substituted with 1 to 5 substituents individually selected from the group consisting of: OH, halogen, cyano and -alkoxy, iv) - C (O) -C1-6-alkyl, wherein C1-6-alkyl is unsubstituted or substituted with 1 to 5 substituents individually selected from the group consisting of: OH, halogen, cyano and C1-6-alkoxy, v) -C O) O-C1-6-alkyl, wherein C1-6-alkyl is unsubstituted or substituted with 1 to 5 substituents individually selected from the group consisting of: OH, halogen, cyano and C1-6-alkoxy, vi) cycloalkyl, unsubstituted or substituted with 1 to 5 substituents individually selected from the group consisting of: OH, halogen, cyano and C 1-6 alkoxy, vii) -S (O) 2- (CH 2) q -NR 1 R 14, wherein q is 0 or 1, R 1 and R 11 are each selected from the group consisting of H and C1-6-alkyl 1, or R 1 and R 1 form, together with the nitrogen to which they are attached, a 3- to 7-membered heterocyclyl containing one or two heteroatoms individually selected from N, O and S, and the heterocyclyl is unsubstituted or substituted by 1 to 5 substituents individually selected from the group consisting of oxo, halogen, C1-6-alkyl and C1-6 -alkoxy, viii) - (CH2) r-NRiiiRiv, where 1, 2 or 3, R1 and Riv are each selected from groups consisting of H and C1-6-alkyl, or R1 and R1 form, together with the nitrogen to which they are attached, a 3- to 7-membered heterocyclyl containing one or two heteroatoms individually selected from N, O and S, and the heterocyclyl is unsubstituted or substituted by 1 to 5 substituents individually selected from the group consisting of oxo, halogen, C1-6-alkyl and C1-6-alkoxy, iix) -C (O) (CH2) s-NRvRvi, where 1, 2 or 3, Rv and Rvi are each independently selected from the group consisting of H and C1-6-alkyl, or Rv and Rvi form, together with the nitrogen to which they are attached, a 3- to 7-membered heterocyclyl containing one or two h eteroatom individually selected from N, O and S, and heterocyclyl is unsubstituted or substituted with 1 to 5 substituents individually selected from the group consisting of oxo, halogen, C1-6-alkyl and C1-6-alkoxy, R2 is halogen, R3 is halogen 5-membered heteroaryl, unsubstituted or substituted with (R *) n, each R * being individually selected from the group consisting of: halogen, C1-6-alkyl, halogen-C1-6-alkyl and hydroxy-C1-6- alkyl, and wherein yen = 1, 2 or 3, and two adjacent R * may form a ring of 4, 5, 6 or 7 C, or a pharmaceutically acceptable salt thereof. |
| priorityDate | 2010-05-10-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
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Total number of triples: 43.