abstract |
The present invention relates to the use of novel LUPANIC DERIVATIVES OF GENERAL FORMULA (I) AND (II), OR OF THE SUBSEQUES, CRYSTALS, COMPLEXES, HYDRATES, OR PHARMACEUTICALLY ACCEPTABLE HYDROLYSATABLE ESTERS, TO PREVENT AND / OR INHIBIT THE GROWTH OF TUMORS AND TO TREAT CANCER OR OTHER PROLIFERATIVE DISEASES, PARTICULARLY TO TREAT LEUKEMIA, LIVER CANCER, UTERUS COLOSS, COLON AND PROSTATE CANCER. The present invention further describes the synthesis of these derivatives and the pharmaceutical formulations which contain them. |