http://rdf.ncbi.nlm.nih.gov/pubchem/patent/PL-80394-B1
Outgoing Links
| Predicate | Object |
|---|---|
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D243-24 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/B65B51-06 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D243-16 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/B65B51-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D243-26 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D243-18 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D243-24 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D243-28 |
| filingDate | 1969-11-25-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationDate | 1975-08-30-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | PL-80394-B1 |
| abstract | 1297629 Benzodiazepines SCHERICO Ltd 21 Nov 1969 [26 Nov 1968 25 June 1969] 57058/69 Heading C2C Compounds of the general formula (X = H, halogen, CF 3 , NO 2 , OH, C 1-6 alkyl or alkoxy; R 1 = C 1-6 alkyl or polyfluoroalkyl, phenyl-(C 1-6 alkyl), C 3-6 cycloalkyl, C 3-6 cycloalkyl-(C 1-6 alkyl), C 2-6 alkenyl, C 1-6 aminoalkyl, C 1-6 alkylamino-(C 1-6 alkyl), di-(C 1-6 alkyl). amino-(C 1-6 alkyl); R 2 = H, C 1-6 alkyl or alkanoyloxy, OH; R 3 = X-Ph, naphthyl, thienyl, pyrryl; R 4 = H, C 1-6 alkyl, (CH 2 ) 2,3 -NR 5 R 6 wherein R 5,6 = H, C 1-6 alkyl), their 4-oxides and acid addition salts thereof are prepared by (a) treating a compound of the formula with a base, (b) subjecting a compound of the formula (L = free or blocked amino group) to intramolecular condensation or (c) reacting a compound of the formula with R 3 MgHal (Hal = halogen), followed by hydrolysis and dehydration, and optionally followed in each case by etherification, oxidation and/or salt formation. The above compounds are tranquillizers, anxiolytics, anticonvulsants and muscle-relaxants, and may be administered in the form of pharmaceutical preparations containing them in association with a carrier.n[GB1297629A] |
| priorityDate | 1968-11-26-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 49.