abstract |
1 Hydrogen monocyclic benzamide 4 - (armnomethyl) piperidine in the formula (I) in which R 1 is methoxy, R 2 is hydrogen, methyl or methoxy, R 3 is hydrogen or batho-chlorine, R 4 is hydrogen or b-methyl alkyl, R 5 is hydrogen, L is C 3- C 6, L is C 3- C 6 , C 2-4 aalkyl, propenyl, C 1 -C 2a lkoxy C 2-3a lkyl, C 1 -C 2a lkyl, C 1 -C 2a lkyl, C 2-3alkylsubstituted hydroxyl group, cyanopropyl, methylcarbonylpropyl, ethoxycarbonylopropyl, dipropylaminocarbonyl propyl, pyrrolidyl propyl, pyrrolidyl pyrrolidyl C 1-C 3a alkyl, 6 - oxy - 3 - chloro-pyridazinyl - C 2- C 3a alkyl, ethylp radical-substituted (c-4), propyl-substituted in formula (c-1), where R 13 is ethyl, ethyl-substituted radical in formula (c-3), where R 13 is ethyl, methylsulfonylamino-methyl, 2-methyl-1, 3-dioxol - 2 - quantity - propyl, oxane - C 1- C 2a lkyl, or bdioxolanomethyl, its stero-isomeric form, N - oxide form or bpharmaceutically acceptable additive acid or base PL PL PL |