abstract |
REFERS TO AN ENCAPSULATED COMPOSITION USING GELATIN, INCLUDING FROM 10 mgA TO 300 mgA OF SERTHRALINE OR A SALT OF SERTHRALINE; AND A VEHICLE IMMISCIBLE IN WATER WHICH IS LIQUID AT 37�C AND MAY BE a) MONO-, DI- � TRIGLYCERIDE, WITH A C4-C18 ACIL GROUP, b) A VEGETABLE OIL SELECTED FROM CORN OIL, PEANUT OIL, SESAME; c) A SURFACTANT OR EMULSATOR SELECTED FROM POLYSORBATE 80, NONYLPHENOXYPOLYOXYETHYLENE, SODIUM DIOCYLSULFOSUCCINATE, AMONG OTHERS; d) A FATTY ACID SELECTED FROM CAPRYLIC ACID, CAPRIC ACID, LAURIC ACID, OLEIC ACID OR LINOLEIC ACID; e) LIQUID ESTER OF AN ALCOHOL AND AN ACID, SELECTED FROM PROPYLENE GLYCOL ESTER OF CAPRYLIC OR CAPRIC ACIDS; f) AN ALCOHOL SELECTED FROM POLYETHYLENE GLYCOL, GLYCERIN, ETHANOL OR PROPYLENE GLYCOL. THIS COMPOSITION ALLOWS TO REACH PEAK LEVELS IN BLOOD IN A LESS TIME |