abstract |
IT REFERS TO A PREPARATION OF A SOFT CAPSULE THAT INCLUDES a) CYCLOSPORINE, AS AN ACTIVE INGREDIENT; b) POLYETHYLENE GLYCOL OR PROPYLENE CARBONATE OR ITS MIXTURE; c) ONE OR A MIXTURE OF ESTERIFIED COMPOUNDS OF FATTY ACID AND PRIMARY ALCOHOL, TRIGLYCERIDE OF MEDIUM CHAIN FATTY ACID, IN PARTICULAR CAPRILIC ACID OR CAPROIC ACID AND A MONOGLYCERIDE OF FATTY ACID IN PARTICULAR OLEIC ACID; d) SURFACTANT THAT HAS A HLB VALUE (HYDROPHILIC-LIPOPHILIC BALANCE) FROM 8 TO 17; THEY ARE PRESENT IN THE PROPORTION OF 1: 0.1-10: 1-10: 1-10 BASED ON WEIGHT |