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publicationDate 2015-06-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber PE-20150722-A1
titleOfInvention MODULATORS OF THE EXPRESSION OF ANDROGENIC RECEPTORS THAT INCLUDE A MODIFIED OLIGONUCLEOTIDE
abstract THE INVENTION REFERS TO COMPOUNDS TARGETING A HUMAN ANDROGEN RECEPTOR (RA) TO INHIBIT THE LEVELS OF THE ANDROGEN RECEPTOR IN A CELL, FOR WHICH THEY ARE USEFUL IN THE TREATMENT OF CANCER AND AS INHIBITORS OF THE GROWTH OR CANCER PROLIFERATION. THE COMPOUNDS OF THE INVENTION INCLUDE A MODIFIED OLIGONUCLEOTIDE WITH A LENGTH OF 10 TO 30 UNITED NUCLEOSIDES. IT ALSO REFERS TO COMPOSITIONS THAT INCLUDE SUCH COMPOUNDS, OPTIONALLY TOGETHER WITH AN ANTIANDROGENIC AGENT, SUCH AS ABIRATERONE, AMONG OTHERS
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