abstract |
REFERRING TO A DOSAGE FORM AS A MICROCAPSULE THAT INCLUDES A CORE OF (A) AN ACTIVE SUBSTANCE OF ACID N- (2- (2-PHTHALIMIDO-ETOXY) -ACETYL) -L-ALANIL-D-GLUTAMICO AND A POLYSACARIDE AS PECTIN OR ALGINATE AND A SLIPPER SUCH AS A CALCIUM OR MAGNESIUM STEARATE, AMONG OTHERS; (B) AN INTERNAL COATING SUCH AS METHACRYLIC ACID COPOLIMER, HYDROXY-PROPYL-METHYL-CELLULOSE PHTHALATE, CELLULOSE ACETATE PHTHALATE, AMONG OTHERS; (C) AN EXTERNAL COATING SUCH AS EUDRAGIT L-55 POLYMER, TALC, AND TRIETHYL CITRATE. SAID ACTIVE COMPOSITION TO THE ILEUS, CEECUS AND COLON, AND IS ADMINISTERED FROM 10 TO 1000 mg IN ONE OR MORE DOSE |