abstract |
THIS INVENTION REFERS TO DIHYDROBENZO DERIVATIVES [B] [1,4] DIAZEPIN-2-ONA OF GENERAL FORMULA I WHERE R1, R2, XEY ARE AS DEFINED IN THE SPECIFICATION AND R3 IS AN AROMATIC HETEROCICLE OF SIX MEMBERS WHICH CONTAINS 1 TO 3 NITROGEN ATOMS OR A PYRIDINE-N-OXIDE SO THAT IT IS ALSO DEFINED IN THE SPECIFICATION. THE INVENTION ALSO REFERS TO MEDICINES CONTAINING THESE COMPOUNDS, A PROCESS FOR ITS PREPARATION AS WELL AS ITS USE FOR THE PREPARATION OF MEDICINES FOR THE TREATMENT OR PREVENTION OF CHRONIC AND / OR ACUTE NEUROLOGICAL DISORDERS. |