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assignee http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_1bde28565d28f037e78bf4a67776ee24
classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D498-04
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-20
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-00
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D498-04
filingDate 2004-09-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_7de096da3e6ed56ec31c64724e0083c1
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_02a02a19757b09826fc9edcc59ae2d0d
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c75f07838a8a23c74523afb6436a2ab3
publicationDate 2009-11-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber NZ-545178-A
titleOfInvention Method for the manufacture of the gaboxadol compound 4,5, 6,7-tetrahydroisoxazolo[5,4-c9]pyridin-3-ol (THIP)
abstract The disclosure relates to a method of preparing gaboxadol compound 4, 5, 6, 7-tetrahydroisoxazolo[5,4-c9]pyridin-3-ol (THIP) useful in the treatment of sleeping disorders. In particular a method of preparing THIP comprising reacting a compound of formula (8b) wherein the substituents are defined in the specification or a salt thereof with an acid, typically a mineral acid, to obtain THIP as an acid addition salt. The present disclosure also relates to several intermediates.
priorityDate 2003-09-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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