http://rdf.ncbi.nlm.nih.gov/pubchem/patent/NZ-517620-A

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filingDate 2000-08-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c2daa97b1b779b5fcf01f63bacc0a156
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_f91c95c215b652d0dc00318c41671087
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publicationDate 2004-02-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber NZ-517620-A
titleOfInvention A conjugate comprising a non-peptide moiety, a linking unit and a cytostatic radical
abstract A conjugate comprises a non-peptide moiety binding to aVb3 or aVb5 integrin (vitronectin) receptors, a linking unit, which can be cleaved enzymatically or hydrolytically with release of the cytotoxic radical or of the radical of a cytostatic or of a cytostatic derivative, and a cytostatic radical or a radical of a cytostatic or of a cytostatic derivative. Preferably the cytostatic radical is camptothecin or 9-aminocamptothecin. The conjugate can be used in the manufacture of a medicament for the treatment of carcinomatous disorders. Also described is process for preparing the conjugates.
priorityDate 1999-09-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 457.