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filingDate 1999-12-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2004-02-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber NZ-511937-A
titleOfInvention Methods and compositions for targeting an activated vitronectin receptor with a ligand comprising adenovirus-2 penton base or fragment thereof
abstract Disclosed are ligands that can selectively bind to activated alpha v beta 3 integrin. A monovalent ligand- mimetic (WOW-1 Fab) which includes a single alpha v integrin-binding domain from multivalent adenovirus penton base is provided. Further disclosed are particular compositions of activated alpha v beta 3-specific ligands, such as an antibody which immunoreacts preferentially with activated alpha v beta 3 integrin. Also described are methods using an activated alpha v beta 3-specific ligand for diagnostic detection of activated alpha v beta 3 integrin in tissues and for the targeted delivery of therapeutic agents to tissues containing activated alpha v beta 3 integrin.
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