http://rdf.ncbi.nlm.nih.gov/pubchem/patent/NO-961169-L
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_94ff2d78578d95d1e8d3a2233c76188d |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D309-30 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D309-32 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07J41-0011 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07J41-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07J51-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-00 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07J41-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07J51-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-704 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D309-32 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P9-00 |
| filingDate | 1996-03-22-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_bb40b469dbcbdf0d334672f29a5b73ab http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_f32a9098ab6a30e5a2a03eb4b3d40ef0 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_51e89757e77668fdc9766f2e4fab66d2 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_3eb3cf1e6a397e8680b27890ad6d5f25 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_6a2559894c01115863e408e79fda3643 |
| publicationDate | 1996-05-24-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | NO-961169-L |
| titleOfInvention | New deoxy and oxygen-substituted sugary 14-aminosteroid compounds |
| abstract | Deoxy and oxygen-substituted sugar-containing 14-amino steroid compounds and the pharmaceutically acceptable acid salts or esters thereof of general formula (I), wherein a) R1 is (i) COOR5, wherein R5 is a 1-6 carbon lower alkyl group, a 1-6 carbon lower alkyl group substituted with an amino group, an arylalkyl or heteroarylalkyl group or a carbocyclic ring, or (ii) CHR6OH where R6 is a hydrogen atom or a 1-6 carbon lower alkyl group, or (iii) COR '' where R ' '' is hydrogen, 1-6 carbon lower alkyl, 1-6 carbon lower alkyl-substituted amino, amino or dialkylamino, and b) R2 is -NR7R8, where R7 and R8, which may be the same or different, are hydrogen atoms or 1 -6 carbon lower alkyl group, and c) R3 is (i) a deoxy or oxygen substituted monosaccharide sugar residue, (II) wherein R9a, R9, R10 and R10a <which may be the same or different are 1-6 carbon lower alkyl, hydrogen, hydroxy, fluoro, alkoxy, acetoxy, arylalkyloxy or benzoxy, Rn is 1-6 carbon lower alkyl, hydrogen, hydroxy, fluoro, benzoxy, arylalkyloxy, heteroarylalkyloxy, acetoxy or alkoxy, wherein further when R 5 is 1-6 carbon lower alkyl, neither R 9, R 10 nor R n can be hydroxy or acetoxy, further provided that when R 9 is hydrogen and R 9 is hydrogen, hydroxy or acetoxy, and R n is hydroxy, acetoxy or alkoxy, R 10 cannot be hydroxy or acetoxy and R 12 is methyl, acetoxymethyl or hydroxymethyl, t may be a single bond or double bond, or (ii) a deoxy or oxygen substituted monosaccharide sugar residue, (III) wherein R n is arylalkyloxy, heteroarylalkyloxy or 1-6 carbon lower alkyl substituted oxosilane and R 12 is methyl and d) R 4 is (i) OH, or (ii) H , or (iii) OR13, where R13 is a monosaccharide sugar residue, acetoxy, benzoxy, arylalkyl or heteroarylalkyl, and e) Z is (i) -CH- where a and b are single bonds, or (ii) = C where either a or b is a double bond. |
| priorityDate | 1993-09-24-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 39.