http://rdf.ncbi.nlm.nih.gov/pubchem/patent/NO-20065948-L

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filingDate 2006-12-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_ec6175c2d33790a4b6a6a5f2868618dc
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publicationDate 2007-01-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber NO-20065948-L
titleOfInvention Quinazolin-4-yl-piperidine and cinnolin-4-yl-piperidine derivatives as PDE10 inhibitors for the treatment of CNS disorders
abstract New piperidyl-substituted quinazoline and isoquinoline derivatives of formula I are disclosed which act as effective phosphodiesterase (PDE) inhibitors. The invention also relates to compounds which are selective inhibitors of PDE 10. The invention further relates to intermediates for the preparation of such compounds; pharmaceutical materials comprising such compounds, and the use of such compounds in methods for treating certain central nervous system (CNS) disorders or other disorders.
priorityDate 2004-07-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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