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filingDate 2005-04-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2005-06-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber NO-20051833-L
titleOfInvention 4- (3,5-dicyanophenoxy) pyrazole derivatives for use as transcriptase modulators in the treatment of IA HIV.
abstract Pyrazole derivatives of formula (I) and pharmaceutically acceptable salts, solvates or derivatives thereof are disclosed. Further described are the use of the compounds in medicine, preparations containing compounds, processes for the preparation of these compounds, as well as intermediates for use in these processes. The described compounds bind to the enzyme reverse transcriptase and are modulators and in particular inhibitors thereof. Reverse transcriptase is implicated in the infectious life cycle of the human immunodeficiency virus (HIV). Compounds that interfere with the function of this enzyme have shown utility in the treatment of conditions caused by HIV and genetically related retroviruses such as acquired immunodeficiency syndrome (AIDS).
priorityDate 2002-09-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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