abstract |
THE PRESENT INVENTION RELATES TO IMIDA:ZOLE DERIVATIVES OF THE GENERAL FORMULA WHEREIN R1, R2, R3 AND R4 ARE AS DEFINED IN THE DESCRIPTION AS WELL AS PHARMACEUTICALLY ACCEPTABLE SALTS AND PROCESSES FOR THE PREPARATION THEREOF. THE INVENTION ALSO RELATES TO MEDICAMENTS CONTAINING SAID IMIDAZOLE DERIVATIVES AND TO THEIR USE FOR THE MANUFACTURE OF MEDICAMENTS FOR THE TREATMENT AND PREVENTION OF MGLUR5 RECEPTOR MEDIATED DISORDERS SUCH AS ACUTE AND/OR CHRONIC NEUROLOGICAL DISORDERS, IN PARTICULAR ANXIETY, OR FOR THE TREATMENT OF CHRONIC AND ACUTE PAIN. |