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filingDate 2001-12-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2010-06-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber MY-141733-A
titleOfInvention Benzimidazole and pyridylimidazole derivatives as ligands for gabaa receptors
abstract THIS INVENTION RELATES TO BENZIMIDAZOLES, PYRIDYLIMIDAZOLES AND RELATED BICYCLIC HETEROARYL COMPOUNDS, ALL OF WHICH MAY BE DESCRIBED BY OF FORMULA I THE INVENTION IS PARTICULARLY RELATED TO SUCH COMPOUNDS THAT BIND WITH HIGH SELECTIVITY AND HIGH AFFINITY TO THE BENZODIAZEPINE SITE OF GABAA RECEPTORS. THIS INVENTION ALSO RELATES TO PHARMACEUTICAL COMPOSITIONS COMPRISING SUCH COMPOUNDS AND TO THE USE OF SUCH COMPOUNDS IN TREATMENT OF CERTAIN CENTRAL NERVOUS SYSTEM (CNS) DISEASES. NOVEL PROCESSES FOR PREPARING COMPOUNDS OR FORMULA I ARE DISCLOSED. THIS INVENTION ALSO RELATES TO THE USE OF BENZIMIDAZOLES,PYRIDYLIMIDAZOLES AND RELATED BICYCLIC HETEROARYL COMPOUNDS OF FORMULA I IN COMBINATION WITH ONE OR MORE OTHER CNS AGENTS TO POTENTIATE THE EFFECTS OF THE OTHER CNS AGENTS. ADDITIONALLY THIS INVENTION RELATES TO THE USE SUCH COMPOUNDS AS PROBES FOR THE LOCALIZATION OF GABAA RECEPTORS IN TISSUE SECTIONS.
priorityDate 2000-12-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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