http://rdf.ncbi.nlm.nih.gov/pubchem/patent/MY-132049-A
Outgoing Links
Predicate | Object |
---|---|
assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_40a92325286ca98dbffa06d2c67ed064 |
classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-415 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D401-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D401-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D403-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D403-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D- http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K- http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D233-64 |
filingDate | 1995-11-23-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_ed2d8b669a9617937769a7a30003095c http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_93665e3fc9cc00f9d7bc090b3eae1931 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_f09f89979fdb321d187f78260424d318 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_9a304f264371f76fc9d194381d4fa36c |
publicationDate | 2007-09-28-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber | MY-132049-A |
titleOfInvention | Certain 4-aminomethyl-2-substituted imidazole derivatives and 2-aminomethyl-4-substituted imidazole derivatives; new classes of dopamine receptor subtype specific ligands |
abstract | DISCLOSED ARE COMPOUNDS OF THE FORMULA :(FORMULA I)WHEREIN R1 REPRESENTS OPTIONALLY SUBSTITUTED ARYL, HETEROARYL, ARYLALKYL, OR CYCLOALKYL GROUPS; X, Z, AND Y ARE OPTIONALLY SUBSTITUTED NITROGEN OR CARBON ATOMS; R3 AND R4 ARE INORGANIC SUBSTITUTENTS WHICH MAY TOGETHER FORM RING STRUCTURES; M IS ZERO, ONE OR TWO; AND R5 AND R6 ARE ARE ORGANIC OR INORGANIC SUBSTITUENTS; AND THE PHARMACEUTICALLY ACCEPTABLE ADDITION SALTS THEREOF, WHICH COMPOUNDS ARE HIGHLY SELECTIVE PARTIAL AGONISTS OR ANTAGONISTS AT BRAIN DOPAMINE RECEPTOR SUBTYPES OR PRODRUGS THEREOF AND ARE USEFUL IN THE DIAGNOSIS AND TREATMENT OF EFFECTIVE DISORDES SUCH AS SCHIZOPHRENIA AND DEPRESSION AS WELL AS CERTAIN MOVEMENT DISORDES SUCH AS PARKINSONISM. |
priorityDate | 1994-11-23-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 26.