abstract |
THE PRESENT INVENTION RELATES TO COMPOUNDS OF THE FORMULA (I), AND PHARMACEUTICALLY -. ACCEPTABLE SAFTS THEREOF WHICH INHIBIT CARBOXYPEPTIDASEU AND THUS CAN BE USED IN THE PREVENTION AND TREATMENT OF DISEASES ASSOCIATED WITH CARBOXYPEPRIDASE U. IN FURTHER ASPECTS, THE INVENTION RELATES TO COMPOUNDS OF THE INVENTION FOR USE IN THERAPY; TO PROCESSES FOR PREPARATION OF SUCH NEW COMPOUNDS; TO PHARMACEUTICAL COMPOSITIONS CONTAINING AT LEAST ONE COMPOUND OF THE INVENTION, OR A PHARMACEUTICALIY ACCEPTABLE SALT THEREOF, AS ACTIVE INGREDIENT; AND TO THE USE OF THE ACTIVE COMPOUNDS IN THE MANUFACTURE OF MEDICAMENTS FOR THE MEDICAL USE INDICATED ABOVE. |