http://rdf.ncbi.nlm.nih.gov/pubchem/patent/MX-PA05006772-A
Outgoing Links
Predicate | Object |
---|---|
assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_b8be6a6c990669567cc455d32b00535e |
classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D215-38 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P5-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P5-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P35-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P5-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D401-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D405-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D409-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P15-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P15-18 |
classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D401-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P5-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D409-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D215-38 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-47 |
filingDate | 2003-12-16-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_a316342109c748cece0de83d4c3527fc |
publicationDate | 2005-09-08-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber | MX-PA05006772-A |
titleOfInvention | DERIVATIVES OF TETRAHYDROQUINOLINE. |
abstract | The present invention relates to tetrahydroquinoline derivatives having the general formula (1) or a pharmaceutically acceptable salt thereof, wherein R1 and R2 are H or Me; R3 is heterocycloalkyl of 2 to 5 carbon-alkyl atoms of 1 to 4 carbon atoms, heteroaryl of 2 to 5 carbon-alkyl atoms of 1 to 4 carbon atoms, aryl of 6 carbon-alkyl atoms of 1 to 4 carbon atoms, (di) alkylaminocarbonylamino of 1 to 4 carbon atoms-alkyl of 2 to 4 carbon atoms, heterocycloalkylcarbonylamino of 2 to 6 carbon atoms-alkyl of 2 to 4 carbon atoms, R5-alkyl of 2 to 4 carbon atoms or R5-carbonyl-alkyl of 1 to 4 carbon atoms; R4 is heteroaryl of 2 to 5 carbon atoms, aryl of 6 carbon atoms, cycloalkyl of 3 to 8 carbon atoms, heterocycloalkyl of 2 to 6 carbon atoms or alkyl of 1 to 6 carbon atoms and R5 is (di) alkylamino of 1 to 4 carbon atoms, alkoxy of 1 to 4 carbon atoms, amino, hydroxy, arylamino of 6 carbon atoms, (di) alkenylamino of 3 to 4 carbon atoms, heteroaryl of 2 to 5 carbon atoms- alkylamino of 1 to 4 carbon atoms, aryl of 6 carbon atoms-alkylamino of 1 to 4 carbon atoms, (di) [alkoxy of 1 to 4 carbon atoms-alkyl of 1 to 4 carbon atoms] amino, ( di) [alkylamino of 1 to 4 carbon atoms-alkyl of 2 to 4 carbon atoms] amino, (di) [amino-alkyl of 2 to 4 carbon atoms] amino or (di) [hydroxy-alkyl of 2 to 4 carbon atoms] amino. The present invention also relates to pharmaceutical compositions containing said derivatives and the use of these derivatives to regulate fertility. |
priorityDate | 2002-12-20-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 385.