abstract |
Amides of 1H-pyrrolo (3,2-b (pyridine-3-carboxylic acid) which bind to the benzodiazepine site of GABAA receptors are described. Such a compound can be used to modulate the ligand binding to GABAA receptors in vivo and in vitro, and are particularly useful in the treatment of a variety of central nervous system (CNS) disorders in humans, domesticated companion animals, and livestock animals. |