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filingDate 2012-10-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_f395d212728a52250cff9ed31ec8ae87
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publicationDate 2019-09-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber MX-367774-B
titleOfInvention N-ACIL-5,6,7, (8-SUBSTITUTE) -TETRAHYDRO- [1,2,4] TRIAZOLO [4,3-a] CHIRAL PYRAZINES, NOVELTY, AS SELECTIVE NK-3 RECEPTOR ANTAGONISTS; PHARMACEUTICAL COMPOSITION, METHODS FOR USE IN NK-3 RECEPTOR-MEDIATED DISORDERS AND ITS CHIRAL SYNTHESIS.
abstract The present invention relates to novel compounds of formula I: (see Formula) and their use in therapeutic treatments. The invention further relates to a novel chiral synthesis of 5,6,7, (8-substituted) -tetrahydro- [1,2,4] triazolo [4,3-a] pyrazines using N-sp3 protecting groups. The invention also provides intermediates for use in the synthesis of compounds of formula I.
priorityDate 2011-10-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 56.