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filingDate 2016-06-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_4bd7c0e0b5de59ab77b808b587f34337
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publicationDate 2018-05-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber MX-2017016611-A
titleOfInvention TGR5 MODULATORS AND METHODS OF USE OF THE SAME.
abstract The application refers to compounds of formula A: (see Formula) or a salt, solvate, ester, tautomer, amino acid conjugate or metabolite thereof. The compounds of formula A are modulators of TGR5 useful for the treatment of various diseases, including metabolic disease, inflammatory disease, autoimmune disease, heart disease, kidney disease, cancer and gastrointestinal disease.
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