http://rdf.ncbi.nlm.nih.gov/pubchem/patent/MX-2014004057-A

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filingDate 2012-10-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_0018c6303f1b1ec842e02aee6a349f04
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_9104db295b6e93ab726a50987a604880
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publicationDate 2014-08-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber MX-2014004057-A
titleOfInvention N-ACIL-5,6,7, (8-REPLACED) -TETRAHYDRO- [1,2,4] TRIAZOLO [4,3-A] PIRA QUIRAL ZINAS, NOVEDOSAS, AS SELECTIVE ANTAGONISTS OF NK-3 RECEPTOR; PHARMACEUTICAL COMPOSITION, METHODS FOR USE IN DISORDERS MEDIATED BY NK-3 RECEPTOR AND ITS CHIRAL SYNTHESIS.
abstract The present invention relates to novel compounds of the formula I: (see Formula) and their use in therapeutic treatments. The invention further relates to a novel chiral synthesis of 5,6,7, (8-substituted) -tetrahydro- [1,2,4] triazolo [4,3-a] pyrazines using N-sp3 protecting groups. The invention also provides intermediaries for use in the synthesis of compounds of the formula I.
priorityDate 2011-10-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 606.