abstract |
The present invention relates to a series of substituted N-phenyl-bipyrrolidine carboxamides of Formula (I) in which R1, R2, M, N and P are as defined in the specification. MORE SPECIFICALLY, THE COMPOUNDS OF THE INVENTION ARE MODULATORS OF H3 RECEPTORS AND THEREFORE ARE USEFUL AS PHARMACEUTICAL AGENTS, IN PARTICULAR IN THE TREATMENT AND / OR PREVENTION OF VARIOUS DISEASES MODULATED BY H3 RECEPTORS COMPRISING THEM. DISEASES ASSOCIATED WITH THE CENTRAL NERVOUS SYSTEM. FURTHERMORE, THE INVENTION ALSO CONCERNS PROCESSES FOR THE PREPARATION OF SUBSTITUTED N-PHENYL-BIPYRROLIDINE CARBOXAMIDES AND INTERMEDIATES USED THEREFOR. |